Taw qhia rauLarazotide
Larazotide(Inn; tseem hu ua ntawm -1001; acetate "}} nws yog ib txwm hloov pauv thaum lub zog hluav taws xob txhawm rau txhim kho cov khoom siv tshuaj (e {. g {{4 4} solubility, ruaj khov, thiab lwm yam})
LarazotidePuas yog hluavtaws peptide . Nws ua haujlwm zoo li lub zog sib tw thiab thim kev sib tshuam mus rau lawv cov feem ntau kaw lub xeev .
Yuav Npaj Li CasLarazotidenyob rau hauv cov kuab tshuaj sib txawv?
Solubility hauv H2O: 16 {.} 67 mg / ml (21.21 mm;) ultrasonic-pab sib txawv.
Solubility hauv DMSO: 3 {. 2 mg (4.07 lub hli rau kev pab cuam tshuam dulethyl tau cuam tshuam loj rau solubility ntawm cov khoom.
Cov qauv ntawm Larazotide?
Muaj ob daim: dawb alkali CAS: {{{{{{}}}}} Qhov txawv ntawm ob daim ntawv no, nthuav dav hauv qab no:


|
Khoom npe |
Tus lej |
Molecular hnyav |
Molecular Cov Qauv |
So |
Rooj mov |
|
Larazotide |
258818-34-7 |
725.83 |
C32H55N9O10 |
Solubility hauv H2O: 2.5 mg / ml (3.44 hli;) Ultrasonic-plived |
{{01.} illally agent zonulin uttrianisticisticist |
|
2.} antiviral kev ua si |
|||||
|
Larazotide acetate |
881851-50-9 |
785.89 |
C34H59N9O12 |
Nws yog me ntsis soluble hauv dej |
1.} artificial hluavtaws peptide |
|
2. Nws ua ncaj qha rau ntawm cov hnyuv mucosa, txo plab thiab kev mob plab zom mov |
Muaj peev xwm tsis muaj khoomLarazotidemuab tau?
Nco ntsoov, nws raug nquahu kom npaj lub diluted ua hauj lwm lim nrog rau ib tug 0}}}}} {1} {1} {1} {1} {1} {1}. pa cawv thiab kev daws kev daws teeb meem yog tseeb.
Nyob rau hauv lub xeev ntshiab, tsis muaj nag dej yuav tsum tau pom nyob rau hauv lub tshuab tsom . Tsis txhob sterilize ntawm qhov kub siab lossis siab}
Cov txiaj ntsig ntawm Larazotide hmoov
{{01.} Hauv cov chaw kuaj mob, Larazotide tau qhia qee lub peev xwm, tshwj xeeb yog cov neeg mob uas haus lub ntsej muag zoo nkauj.
1) Larazotide tuaj yeem daws cov tsos mob plab zom mov xws li mob plab, mob plab thiab raws plab
2) Nws tuaj yeem txo qhov nce hauv plab hnyuv tso cai tshwm sim los ntawm gluten thiab txo txoj kev pheej hmoo ntawm mucosal kev puas tsuaj.
2.} kev cai ntawm autoimmunity
Larazotidetsis ncaj ncees inhibits qhov kev tsim cov khoom siv los ntawm kev txo qis ntawm cov txheej txheem autoivcator, txo qis kev pheej hmoo carbonation celiaimmune puas .

Phiv los ntawmLarazotide hmoov
Cov kev mob tshwm sim yuav tsum tau piav qhia los ntawm peb lub ntsiab lus hauv qab no
1. Cov kev mob tshwm sim muaj qhov mob plab, mob plab zom mov, mob plab, mob taub hau thiab kiv taub hau}
2. Cov kev mob tshwm sim muaj tshwm sim tsis tshua muaj, tab sis lawv tseem yuav tsum ua kev ua xua thiab ua pa tawm ntawm kev ua xua tam sim ntawd .
3. pawg pawg yuav tsum ceev faj tshwj xeeb, suav nrog cov poj niam cev xeeb tub, ua kom cov menyuam yaus tsis muaj lactive {{2 2}}
Phau ntawv
1.https: // doi {{. org / 10.1111 / j .1749-6632.2012.06538. x
2.https: // pubmed . NCBi . ni}} gov / 25724700 /
3https: // . sagepub {}} com / doi / full / 10.119884819868235




